Risperidone Raw Powder CAS. 106266-06-2 99% Ubunyulu

Ingcaciso yeMveliso
I-Risperidone, i-molecular formula c23h27fn4o2, igama lekhemikhali 3 - [2 - [4 - (6-fluoro-1,2-benzoisoxazole-3-yl) - 1-piperidyl] ethyl] - 6,7,8,9-tetrahydro-2-methyl-4h-pyrido [1,2] i-pyrido esetyenzisiweyo, i-dianechrid, i-adine, i-adine, i-pyrido esetyenzisiweyo ukunyanga i-schizophrenia ebukhali kunye nengapheliyo. Ngokukodwa kwiimpawu ezintle nezimbi kunye neempawu zeemvakalelo ezinxulumene nazo (ezifana nokuxhalaba, ukudakumba, njl.). Kwakhona kunokunciphisa iimpawu zeemvakalelo ezinxulumene ne-schizophrenia. Kwizigulane ezinonyango olusebenzayo kwisigaba esibuhlungu, le mveliso inokuqhubeka nokusebenzisa iklinikhi yayo kwisigaba sokugcina.
I-COA
| IZINTO | UMGANGATHO | ISIPHUMO SOVAVANYO |
| Isivavanyi | 99% | Iyahambelana |
| Umbala | Umgubo omhlophe | Iyahambelana |
| Ivumba | Akukho vumba likhethekileyo | Iyahambelana |
| Ubungakanani besuntswana | I-100% iphumelele i-80mesh | Iyahambelana |
| Ilahleko ekomisweni | ≤5.0% | 2.35% |
| Intsalela | ≤1.0% | Iyahambelana |
| Intsimbi enzima | ≤10.0ppm | 7ppm |
| As | ≤2.0ppm | Iyahambelana |
| Pb | ≤2.0ppm | Iyahambelana |
| Intsalela yesitshabalalisi | Ibi | Ibi |
| Ubalo lweepleyiti lulonke | ≤100cfu/g | Iyahambelana |
| Igwele kunye noMngundo | ≤100cfu/g | Iyahambelana |
| E.Coli | Ibi | Ibi |
| Salmonella | Ibi | Ibi |
| Ukuqukumbela | Qhagamshelana neNgcaciso | |
| Ugcino | Igcinwe kwindawo epholileyo kunye neyomileyo, zigcine kude nokukhanya okuqinileyo kunye nobushushu | |
| Beka ubomi kwishelufa | Iminyaka emi-2 xa igcinwe ngokufanelekileyo | |
Umsebenzi
Inyathelo 1 Zolile
I-Risperidone ivelisa umphumo wokuthomalalisa ngokulawula ukulingana kwee-neurotransmitters kwingqondo ukunciphisa umsebenzi wobuchopho ogqithiseleyo.
2. I-Antipsychotic
I-Risperidone iyakwazi ukuvala i-dopamine D2 receptors, ukunciphisa umsebenzi we-dopamine, kunye nokunciphisa iimpawu ezintle ezifana nemibono kunye nokukhohlisa.
3. Amachiza okudakumba
I-Risperidone inokuphucula ukungasebenzi kokuhanjiswa kweemvakalelo, inyuse amanqanaba e-serotonin kunye ne-norepinephrine, kwaye ithobe ukudakumba.
4. Yeka ukugabha
I-Risperidone ingasetyenziselwa njenge-peripheral opioid receptor antagonist kwinkqubo ye-nervous central kwaye inomphumela othile we-antiemetic.
5. Iprolactin inhibition
I-Risperidone inokukhuphisana ngokunqanda i-hypothalamic prolactin ekhupha into, ekhokelela ekunciphiseni ukukhutshwa kweprolactin.
I-Risperidone isetyenziswa ikakhulu kunyango lwe-schizophrenia kunye nokuphazamiseka okunxulumene noko. Kuyimfuneko ukunikela ingqalelo ekubekeni iliso kwiziphumo ebezingalindelekanga ezifana ne-bradykinesia kunye nokuqunjelwa xa usebenzisa i-risperidone, kwaye ulandele isikhokelo sikagqirha ukulungelelanisa umthamo.
Isicelo
Ukusetyenziswa kwe-risperidone powder kwiinkalo ezahlukeneyo ikakhulu kubandakanya le miba ilandelayo:
1. Unyango lwesigulo sengqondo : I-Risperidone sisiyobisi se-antipsychotic sesizukulwana sesibini esisetyenziswa ikakhulu ukunyanga i-schizophrenia. Inokuphucula ngokufanelekileyo iimpawu ezintle ze-schizophrenia (ezifana nemibono, ukukhohlisa, ukuphazamiseka kokucinga) kunye neempawu ezimbi (ezifana nokungaphenduli, ukunganakwa). Ukongeza, i-risperidone inokunciphisa iimpawu zeemvakalelo ezinxulumene ne-schizophrenia, njengokudakumba, ukuxhalaba, njl.
2. I-bipolar disorder : I-Risperidone isetyenziselwa ukunyanga ingxaki ye-bipolar, ngakumbi i-manic episodes, ukuzinzisa isimo sengqondo kunye nokuphucula isimo sengqondo.
3. Okunye ukuphazamiseka kwengqondo : i-risperidone kwi-obsessive-compulsive disorder, i-anxiety disorder disorder, i-hyperactive tic disorder nayo inesicelo esithile, i-clinical efficacy.
4. I-AutismI-Risperidone inokusetyenziswa kwezinye iimeko ukunyanga ukucaphuka kunye nokuziphatha okundlongondlongo okuhambelana noluphazamiseko.
Iimveliso ezinxulumeneyo
Umzi-mveliso omtsha oluhlaza ukwabonelela ngeeAmino acids ngolu hlobo lulandelayo:
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