●Yintoni i I-Synephrine Hydrochloride?
I-Synephrine HCl yindlela ye-hydrochloride ye-synephrine, kunye ne-chemical formula C₉H₁₃NO₂·HCl (i-molecular weight 203.67). I-precursor yayo yendalo ye-synephrine ifumaneka ikakhulu kwiziqhamo ezincinci ezomileyo (i-citrus aurantium) yesityalo se-Rutaceae. I-Citrus aurantium isasazwe ngokubanzi kumaphondo e-Yangtze River Basin yase-China, njenge-Sichuan, i-Jiangxi, kunye ne-Zhejiang. Umxholo we-synephrine kwiziqhamo zayo ezincinci unokufikelela kwi-30% yesisindo esomileyo. Ukukhutshwa kwemveli kuxhomekeke ekutsalweni kotywala (i-75% ye-ethanol reflux extraction amaxesha ama-3, isivuno ≥ 85%), kodwa kwiminyaka yakutshanje, iteknoloji entsha igxile ekusebenzeni okuluhlaza kunye nokusebenza okuphezulu:
Ukwahlulwa kwe-enzymatic hydrolysis-membrane: i-compound pectinase hydrolyzes pectin kwi-40 ° C kunye ne-pH 4.5, idibene ne-0.22μm ye-inorganic ceramic membrane filtration, izinga lokususa ukungcola lifikelela kwi-91%, kwaye ukucoceka kwanda ukuya ngaphezu kwe-95%;
Iteknoloji yokutshintshwa kwefungal: I-Academy yaseShayina yeSayensi yezoLimo iye yaphuhlisa indlela ye-Ganoderma lucidum fermentation ukuvelisa izinto ezifana ne-synephrine, ukunciphisa iindleko nge-30% kunye nokunciphisa uxinzelelo lokumbiwa kwemigodi ngokungekho mthethweni kwimithombo yasendle.
●Yintoni naIingeneloKwe I-Synephrine Hydrochloride ?
I-Synephrine hydrochloride, njenge-agonist emibini ye-adrenaline α/β receptors, iphinda ihlaziye ixabiso lekliniki ngeziphumo ezininzi ekujoliswe kuzo:
1. I-Cardiovascular Emergency
I-receptors evuyisayo ye-α ukuxinzelela imithwalo yegazi kunye nokwandisa uxinzelelo lwegazi, olusetyenziselwa i-anesthesia, i-hypotension, ukuhlangulwa kokutshatyalaliswa, kunye nesantya sokuqala si-40% ngokukhawuleza kuneziyobisi zendabuko;
Ukuvuselela i-receptors ye-β ukunyusa i-contractility ye-myocardial kunye nokuphucula umsebenzi wokumpompa izigulana ezinokusilela kwentliziyo.
2. Ungenelelo lweNkqubo yokuphefumla
I-Synephrinehidrochlorideunako sI-bronchial ilula kakhulu imisipha egudileyo, ichasene ngokupheleleyo ne-histamine-induced spasm, kwaye yandise i-FEV1 index of lung function kwizigulane ezine-asthma ye-bronchial ngama-25%.
3. Ukulawulwa kweMetabolic
I-fat oxidation revolution: Ukuvuselela isantya se-metabolism ye-brown adipose tissue nge-50%, kunye nokutya kwansuku zonke kwe-20 mg kunokunciphisa izinga lamafutha omzimba nge-3.5%;
I-Neuroprotective potential: I-reversibly inhibit acetylcholinesterase, iphucula amanqaku okusebenza kwengqondo kwizigulane ze-dementia nge-30%, kwaye ubude besenzo buphindwe kabini kumachiza aqhelekileyo.
Ukufunyanwa komda wokuwela imida: Uphononongo luka-2020 olwenziwe yiYunivesithi yaseMazantsi-ntshona luveze okokuqala umsebenzi walo wokugcinwa kweziqhamo kunye nemifuno - 0.1mmol/Lsynephrine hydrochlorideunyango lunokuthintela umsebenzi we-polyphenol oxidase kwi-litchi peel, ukulibazisa umdaka ngokulawula i-membrane ye-lipid metabolism, kunye nokwandisa ubomi beshelufu ukuya kwiintsuku ze-14.
●Yintoni naIsiceloOf I-Synephrine Hydrochloride?
1. IMarike ePhambili kwiNdawo yoShishino
Amalungiselelo oncedo lokuqala: ii-injection kunye neepilisi zisetyenziselwa i-hypotension yokuhlinzwa kunye nokutshatyalaliswa.
Ukulawulwa kwezifo ezingapheliyo: kudibaniswa ne-aminophylline ukunyanga i-asthma ye-bronchial, izinga lokuhlaselwa ngokukhawuleza liyancipha ngama-60%.
Amachiza okunciphisa umzimba: njengento ebambeleyo yendalo ye-ephedrine, inokusetyenziswa njengesongezelelo sezemidlalo.
2. Inguqulelo yoLondolozo lwezoLimo
I-Lychee browning inhibitor: emva kokuba i-lychee ivunwe kwaye iphathwe ngayosynephrine hydrochloride, ixabiso lilonke yi-1/3 kuphela yekhonkco elibandayo eliqhelekileyo.
I-Citrus yokugubungela i-antiseptic: i-nanoemulsion idibaniswe ne-chitosan, izinga lokulwa ne-antibacterial> 99%, kwaye ixesha lokugcinwa kwiqondo lokushisa legumbi landiswa ngeentsuku ezingama-21.
3. Ukwandiswa kweeMveliso zoMthengi eziSebenzayo
Iziphuzo zamandla: "I-Synephrine + taurine" iziphuzo ezisebenzayo zinokuphucula ukunyamezela kwezemidlalo
Ukutya kwempilo ye-Neural: amalungiselelo e-capsule ejolise kwi-acetylcholinesterase ukuphucula ukukhubazeka kwememori kubantu abadala.
● Newgreen Supply High Quality I-Synephrine Hydrochloride Umgubo
Ixesha lokuposa: Jul-18-2025


