Risperidone Raw Powder CAS. 106266-06-2 99% Kuchena

Product Description
Risperidone, molecular formula c23h27fn4o2, zita remakemikari 3 - [2 - [4 - (6-fluoro-1,2-benzoisoxazole-3-yl) - 1-piperidyl] ethyl] - 6,7,8,9-tetrahydro-2-methyl-4h-pyrido [1,2] zvinodhaka-psychrimi, α4, psychrimi, α4, psychrimi yakashandiswa kurapa acute uye chisingaperi schizophrenia. Kunyanya kune zvakanaka uye zvisina kunaka zviratidzo uye zvine chekuita nezviratidzo zvepfungwa (sekufunganya, kuora mwoyo, nezvimwewo). Inogonawo kuderedza zviratidzo zvepfungwa zvine chokuita neschizophrenia. Kune varwere vane kurapa kunoshanda muchikamu cheacute, chigadzirwa ichi chinogona kuenderera mberi nekushandisa kiriniki yayo muchikamu chekugadzirisa.
COA
| ZVINHU | STANDARD | TEST RESULT |
| Assay | 99% | Conforms |
| Color | Upfu chena | Conforms |
| Kunhuwa | Hapana kunhuhwirira kwakakosha | Conforms |
| Chikamu saizi | 100% inopfuura 80mesh | Conforms |
| Kurasikirwa pakuomeswa | ≤5.0% | 2.35% |
| Residue | ≤1.0% | Conforms |
| Heavy metal | ≤10.0ppm | 7ppm |
| As | ≤2.0ppm | Conforms |
| Pb | ≤2.0ppm | Conforms |
| Mushonga wezvipembenene wasara | Negative | Negative |
| Yese plate count | ≤100cfu/g | Conforms |
| Yeast & Mold | ≤100cfu/g | Conforms |
| E.Coli | Negative | Negative |
| Salmonella | Negative | Negative |
| Mhedziso | Ita zvinoenderana neSpecification | |
| Storage | Yakachengetwa munzvimbo Inotonhorera & Yakaoma, Ramba Kure Nechiedza Chakasimba uye Kupisa | |
| Sherufu hupenyu | 2 years pakachengetwa zvakanaka | |
Function
Danho 1 Dzikama
Risperidone inogadzira kudzikamisa mhedzisiro nekudzora kuenzana kwemaurotransmitters muhuropi kuderedza kuwandisa kwehuropi kuita.
2. Antipsychotic
Risperidone inokwanisa kuvhara dopamine D2 receptors, kuderedza dopamine basa, uye kuderedza zviratidzo zvakanaka zvakadai sekufungidzira uye kunyengera.
3. Antidepressants
Risperidone inogona kuvandudza kusagadzikana kwekutapurirana kwemanzwiro, kuwedzera serotonin uye norepinephrine mazinga, uye kuderedza kushushikana.
4. Rega kurutsa
Risperidone inogona kushandiswa seanopikisa opioid receptor antagonist mukati menheyo system uye ine imwe antiemetic mhedzisiro.
5. Prolactin inhibition
Risperidone inogona kukwikwidza inhibit hypothalamic prolactin kuburitsa chinhu, zvichikonzera kuderera kweprolactin secretion.
Risperidone inonyanya kushandiswa kurapa schizophrenia uye zvine chekuita nekukanganisika. Zvakakosha kubhadhara kutarisa zvinogona kuitika zvakadai sebradykinesia uye kuvimbiswa paunenge uchishandisa risperidone, uye kutevera mazano echiremba kuti agadzirise dose.
Application
Kushandiswa kwerisperidone poda munzvimbo dzakasiyana-siyana kunonyanya kusanganisira zvinotevera:
1. Kurapwa kwechirwere chepfungwa : Risperidone mushonga wechizvarwa chechipiri unoshandiswa kurapa schizophrenia. Inogona kuvandudza zvinobudirira zviratidzo zvakanaka zveschizophrenia (zvakadai sekufungidzira, kunyengedza, kukanganisa kufunga) uye zviratidzo zvisina kunaka (zvakadai sokusapindura, kusava nehanya). Mukuwedzera, risperidone inogonawo kuderedza zviratidzo zvepfungwa zvine chokuita neschizophrenia, zvakadai sekuora mwoyo, kufunganya, nezvimwewo.
2. Bipolar disorder : Risperidone inoshandiswa kurapa bipolar disorder, kunyanya manic episodes, kudzikamisa manzwiro nekuvandudza mafungiro.
3. Zvimwe zvirwere zvepfungwa : risperidone in obsessive-compulsive disorder, generalized anxiety disorder, hyperactive tic disorder inewo imwe application, kliniki efficacy.
4. Autism: Risperidone inogona kushandiswa mune dzimwe nguva kurapa kushatirwa uye hukasha maitiro ane chekuita ne autism.
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