●Kodi Ndi Chiyani Synephrine Hydrochloride?
Synephrine HCl ndi mtundu wa hydrochloride wa synephrine, wokhala ndi mankhwala C₉H₁₃NO₂·HCl (mamolekyu olemera 203.67). Kalambulabwalo wake wachilengedwe wa synephrine makamaka amachokera ku zipatso zazing'ono zouma (citrus aurantium) za chomera cha Rutaceae. Citrus aurantium imagawidwa kwambiri m'zigawo za Yangtze River Basin ku China, monga Sichuan, Jiangxi, ndi Zhejiang. Zomwe zili mu synephrine mu zipatso zake zazing'ono zimatha kufika ku 30% ya kulemera kowuma. Kutulutsa kwachikhalidwe kumadalira kutulutsa mowa (75% ethanol reflux m'zigawo katatu, zokolola ≥ 85%), koma m'zaka zaposachedwa, luso laukadaulo limayang'ana kwambiri zobiriwira komanso zapamwamba:
Enzymatic hydrolysis-membrane kulekana: pawiri pectinase hydrolyzes pectin pa 40 ° C ndi pH 4.5, pamodzi ndi 0.22μm inorganic ceramic nembanemba kusefera, ndi zonyansa kuchotsa mlingo kufika 91%, ndi chiyero chawonjezeka kupitirira 95%;
Ukadaulo wolowa m'malo mwa fungal: Bungwe la Chinese Academy of Agricultural Sciences lapanga njira yowotchera ya Ganoderma lucidum kuti ipange zinthu ngati synephrine, kuchepetsa mtengo ndi 30% ndikuchepetsa kukakamizidwa kwa migodi yosaloledwa ya zinthu zakuthengo.
●Ndi ChiyaniUbwinoZa Synephrine Hydrochloride ?
Synephrine hydrochloride, monga agonist wapawiri wa adrenaline α/β zolandilira, amasinthanso phindu lachipatala kudzera muzotsatira zambiri:
1. Matenda a mtima
Zosangalatsa za α zolandilira kuti zichepetse mitsempha yamagazi ndikuwonjezera kuthamanga kwa magazi, komwe kumagwiritsidwa ntchito pochita opaleshoni, hypotension, kupulumutsa kugwedezeka, ndi liwiro loyambira ndi 40% mwachangu kuposa mankhwala azikhalidwe;
Kuyambitsa ma β-receptors kuti apititse patsogolo mgwirizano wa myocardial ndikuwongolera ntchito yopopa ya odwala omwe ali ndi vuto la mtima.
2. Njira Yothandizira Kupuma
Synephrinehhydrochlorideakhoza sImakulitsa kwambiri minofu yosalala ya bronchial, imalepheretsa kufalikira kwa histamine, ndikuwonjezera index ya FEV1 yamapapo kwa odwala omwe ali ndi mphumu ya bronchial ndi 25%.
3. Metabolic Regulation
Kusintha kwamafuta oxidation: Kulimbikitsa kagayidwe kazakudya zamafuta a bulauni ndi 50%, ndipo kudya kwa 20 mg tsiku lililonse kumatha kuchepetsa kuchuluka kwamafuta amthupi ndi 3.5%;
Kuthekera kwa Neuroprotective: Kuletsa mosinthika acetylcholinesterase, kupititsa patsogolo chidziwitso cha odwala omwe ali ndi vuto la dementia ndi 30%, ndipo nthawi yogwira ntchito imakhala yowirikiza kawiri kuposa yamankhwala wamba.
Kupezeka kwa malire: Kafukufuku wa 2020 wochitidwa ndi Southwest University adawulula kwa nthawi yoyamba ntchito yake yosunga zipatso ndi masamba - 0.1mmol/Lsynephrine hydrochlorideKuchiza kumatha kulepheretsa ntchito ya polyphenol oxidase mu peel ya litchi, kuchedwetsa browning mwa kuwongolera kagayidwe ka lipid ka membrane, ndikukulitsa moyo wa alumali mpaka masiku 14.
●Ndi ChiyaniKugwiritsa ntchitoOf Synephrine Hydrochloride?
1. Msika Wopambana M'munda Wamankhwala
Thandizo loyamba kukonzekera: jakisoni ndi mapiritsi ntchito opaleshoni hypotension ndi mantha.
Kasamalidwe ka matenda osachiritsika: kuphatikiza ndi aminophylline pochiza mphumu ya bronchial, chiwopsezo chowopsa chimachepetsedwa ndi 60%.
Mankhwala ochepetsa thupi: monga choloweza mmalo mwachilengedwe cha ephedrine, atha kugwiritsidwa ntchito ngati chowonjezera chamasewera.
2. Agricultural Preservation Innovation
Lychee browning inhibitor: lychee ikakololedwa ndikuthandizidwasynephrine hydrochloride, mtengo wonse ndi 1/3 yokha ya unyolo wozizira wachikhalidwe.
Kupaka kwa citrus antiseptic: nanoemulsion yophatikizidwa ndi chitosan, kuchuluka kwa antibacterial ndi> 99%, ndipo nthawi yosungira kutentha kwa firiji kumakulitsidwa ndi masiku 21.
3. Kuwonjezedwa kwa Zogulitsa Zogwira Ntchito
Zakumwa zamphamvu: "Synephrine + taurine" zakumwa zogwira ntchito zimatha kupititsa patsogolo kupirira kwamasewera
Chakudya chathanzi cha Neural: Kukonzekera kapisozi kolunjika ku acetylcholinesterase kuti apititse patsogolo kuwonongeka kwa kukumbukira kwa okalamba.
● Newgreen Supply High Quality Synephrine Hydrochloride Ufa
Nthawi yotumiza: Jul-18-2025


