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Synephrine Hydrochloride: "Ihe na-eme ka ọbara mgbali elu" ewepụtara na Citrus Aurantium

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Gịnị bụ Synephrine Hydrochloride?

Synephrine HCl bụ hydrochloride ụdị synephrine, na usoro kemịkal C₉H₁₃NO₂ · HCl (molecular arọ 203.67). A na-enweta synephrine sitere n'okike sitere na mkpụrụ osisi mịrị amị (citrus aurantium) nke osisi Rutaceae. A na-ekesa citrus aurantium na mpaghara Yangtze River Basin nke China, dị ka Sichuan, Jiangxi, na Zhejiang. Ọdịnaya synephrine dị na mkpụrụ osisi ya na-eto eto nwere ike iru 30% nke ibu akọrọ. Omenala mmịpụta na-adabere na mmịpụta mmanya (75% ethanol reflux mmịpụta 3 ugboro, mkpụrụ ≥ 85%), mana n'afọ ndị na-adịbeghị anya, ihe ọhụrụ teknụzụ lekwasịrị anya na akwụkwọ ndụ akwụkwọ ndụ na arụmọrụ dị elu:

Enzymatic hydrolysis-membrane nkewa: compound pectinase hydrolyzes pectin na 40 ° C na pH 4.5, jikọtara ya na 0.22μm inorganic seramiiki akpụkpọ anụ filtration, na-adịghị ọcha ọnụego ruru 91%, na ịdị ọcha na-abawanye karịa 95%;

Teknụzụ nnọchi nke fungal: Mahadum China nke Sayensị Ọrụ Ugbo ewepụtala usoro ịgba ụka Ganoderma lucidum iji mepụta ihe ndị dị ka synephrine, na-ebelata ọnụ ahịa site na 30% ma belata nrụgide nke ngwupụta akụ na ụba iwu na-akwadoghị.

Kedu ihe bụUruNke Synephrine Hydrochloride ?

Synephrine hydrochloride, dị ka agonist dual nke adrenaline α / β ndị na-anabata ya, na-emegharị uru ụlọ ọgwụ site na mmetụta dị iche iche:

1. Mberede obi

Ndị na-anabata α na-akpali akpali iji gbochie arịa ọbara ma na-abawanye ọbara mgbali elu, nke a na-eji maka mgbakasị ahụ, hypotension, nnapụta ujo, na mmalite ọsọ ọsọ bụ 40% ngwa ngwa karịa ọgwụ ọdịnala;

Na-eme ka ndị na-anabata β rụọ ọrụ iji kwalite nkwekọrịta myocardial ma melite ọrụ mgbapụta nke ndị ọrịa nwere nkụda obi.

2. Ntinye aka na usoro iku ume

Synephrinehydrochloridenwere ike sna-agbasawanye uru ahụ dị nro nke bronchial nke ọma, na-emegide spasm nke na-akpata histamine kpamkpam, ma na-abawanye ndeksi FEV1 nke ọrụ ngụgụ na ndị ọrịa nwere ụkwara ume ọkụ site na 25%.

3. Metabolic Iwu

Mgbanwe oxidation abụba: kpalie ọnụego metabolic nke adipose anụ ahụ na-acha aja aja site na 50%, na oriri 20 mg kwa ụbọchị nwere ike ibelata ọnụego abụba ahụ site na 3.5%;

Ike Neuroprotective: Na-egbochi acetylcholinesterase na-agbanwe agbanwe, na-emeziwanye ọrụ ọgụgụ isi nke ndị ọrịa dementia site na 30%, na ogologo oge nke ime ihe bụ okpukpu abụọ nke ọgwụ ndị a na-emekarị.

Nchọpụta gafere oke: Nnyocha 2020 sitere na Mahadum Southwest kpughere na nke mbụ ọrụ nchekwa mkpụrụ osisi na akwụkwọ nri ya - 0.1mmol/Lsynephrine hydrochlorideọgwụgwọ nwere ike igbochi ọrụ nke polyphenol oxidase na litchi bee, na-egbu oge browning site na-achịkwa akpụkpọ ahụ lipid metabolism, na ịgbatị ndụ shelf ruo ụbọchị 14.

 

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Kedu ihe bụNgwaOf Synephrine Hydrochloride?

1. Ahịa Na-achị Na-ahụ Maka Ọgwụ Na-ahụ Maka Ọgwụ

Nkwadebe enyemaka mbụ: a na-eji injections na mbadamba ihe maka ịwa ahụ hypotension na ujo.

Nlekọta ọrịa na-adịghị ala ala: jikọtara ya na aminophylline iji gwọọ ụkwara ume ọkụ nke bronchi, ọnụ ọgụgụ ọgụ dị ukwuu na-ebelata site na 60%.

Ọgwụ na-ebelata ibu: dị ka ihe eji dochie anya ephedrine, enwere ike iji ya dị ka mgbakwunye egwuregwu.

2. Agricultural ichekwa Innovation

Lychee browning inhibitor: mgbe ewechara lychee ma mesoo yasynephrine hydrochloride, ngụkọta ọnụ ahịa bụ nanị 1/3 nke omenala oyi yinye.

Citrus antiseptik mkpuchi: nanoemulsion jikọtara ya na chitosan, ọnụego nje nje> 99%, na oge nchekwa na ụlọ okpomọkụ na-agbatị ụbọchị 21.

3. Mgbatị nke ngwaahịa ndị ahịa na-arụ ọrụ

Ihe ọṅụṅụ ike: "Synephrine + taurine" ihe ọṅụṅụ na-arụ ọrụ nwere ike imezi ntachi obi egwuregwu

Nri ahụike akwara: nkwadebe capsule na-ezubere acetylcholinesterase iji kwalite mmetụ ebe nchekwa na ndị agadi.

● Ọdịmma nke Newgreen Supply Synephrine Hydrochloride Ntụ ntụ

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Oge nzipu: Jul-18-2025