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Synephrine Hydrochloride: "Abin da ke Haɓaka Hawan Jini na Halitta" An Cire Daga Citrus Aurantium

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Menene Synephrine Hydrochloride?

Synephrine HCl shine nau'in hydrochloride na synephrine, tare da tsarin sinadaran C₉H₁₃NO₂ · HCl (nauyin kwayoyin 203.67). Sinephrine na asali na dabi'a ya samo asali ne daga busassun 'ya'yan itatuwa masu tasowa (citrus aurantium) na shuka Rutaceae. Citrus aurantium yana bazuwa a kogin Yangtze na kasar Sin, kamar su Sichuan, Jiangxi, da Zhejiang. Abubuwan da ke cikin synephrine a cikin ƙananan 'ya'yan itatuwa na iya kaiwa zuwa 30% na nauyin busassun. Haɗin al'ada ya dogara ne akan hakar barasa (75% ethanol reflux hakar sau 3, yawan amfanin ƙasa ≥ 85%), amma a cikin 'yan shekarun nan, ƙirar fasaha ta mai da hankali kan kore da ingantaccen inganci:

Enzymatic hydrolysis-membrane rabuwa: fili pectinase hydrolyzes pectin a 40 ° C da pH 4.5, hade tare da 0.22μm inorganic yumbu membrane tacewa, da ƙazanta adadin ya kai 91%, da kuma tsarki ya karu zuwa fiye da 95%;

Fasahar canza kayan aikin fungal: Cibiyar Nazarin Kimiyyar Aikin Noma ta kasar Sin ta samar da wata hanyar fermentation ta Ganoderma lucidum don samar da sinadarai masu kama da synephrine, rage farashi da kashi 30% da kuma rage matsin lamba na hakar albarkatun daji ba bisa ka'ida ba.

Menene TheAmfaniNa Synephrine Hydrochloride ?

Synephrine hydrochloride, a matsayin mai dual agonist na adrenaline α / β masu karɓa, yana sake fasalin darajar asibiti ta hanyar tasiri mai yawa:

1. Gaggawa na Zuciya

Masu karɓa na α masu ban sha'awa don ƙaddamar da jini da kuma ƙara yawan karfin jini, wanda ake amfani dashi don maganin sa barci, rashin jin dadi, ceton girgiza, da saurin farawa shine 40% sauri fiye da magungunan gargajiya;

Kunna masu karɓar β don haɓaka ƙaƙƙarfan ƙwayar zuciya da haɓaka aikin famfo na marasa lafiya tare da gazawar zuciya.

2. Tsangwama Tsarin Numfashi

Synephrinehydrchlorideiya ssosai dilate bronchial santsi tsoka, gaba daya antagonize histamine-induced spasm, da kuma ƙara FEV1 index na huhu aiki a marasa lafiya da Bronchial fuka da 25%.

3. Tsarin Halitta

Juyin Juyin Halittar Fat: Ƙarfafa yawan adadin ƙwayar adipose mai launin ruwan kasa da kashi 50%, kuma shan 20 MG na yau da kullun na iya rage yawan kitsen jiki da 3.5%;

Ƙimar Neuroprotective: Maimaituwa yana hana acetylcholinesterase, inganta aikin fahimi na marasa lafiya da 30%, kuma tsawon lokacin aikin shine sau biyu na kwayoyi na al'ada.

Gano kan iyaka: Binciken 2020 na Jami'ar Kudu maso Yamma ya bayyana a karon farko aikin kiyaye 'ya'yan itace da kayan lambu - 0.1mmol/Lsynephrine hydrochlorideJiyya na iya hana ayyukan polyphenol oxidase a cikin kwasfa na litchi, jinkirta launin ruwan kasa ta hanyar daidaita metabolism lipid membrane, da kuma tsawaita rayuwar shiryayye zuwa kwanaki 14.

 

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Menene TheAikace-aikaceOf Synephrine Hydrochloride?

1. Kasuwa Mai Mahimmanci A Filin Magunguna

Shirye-shiryen taimakon farko: ana amfani da allurai da allunan don hypotension na tiyata da girgiza.

Gudanar da cututtuka na yau da kullum: haɗe tare da aminophylline don magance asma na bronchial, an rage yawan mummunan harin da kashi 60%.

Magungunan asarar nauyi: azaman madadin halitta don ephedrine, ana iya amfani dashi azaman kari na wasanni.

2. Kirkirar Kiyaye Noma

Lychee browning inhibitor: bayan an girbe lychee kuma an bi da shisynephrine hydrochloride, jimlar farashin shine kawai 1/3 na sarkar sanyi na gargajiya.

Citrus maganin antiseptik shafi: nanoemulsion hade da chitosan, da antibacterial rate ne> 99%, da kuma ajiya lokaci a dakin zafin jiki da aka tsawaita da 21 kwanaki.

3. Tsawaita Kayayyakin Masu Amfani

Abubuwan sha na makamashi: "Synephrine + taurine" abubuwan sha masu aiki na iya inganta juriyar wasanni

Abincin lafiyar jijiyoyi: shirye-shiryen capsule da ke niyya ga acetylcholinesterase don inganta ƙwaƙwalwar ƙwaƙwalwa a cikin tsofaffi.

● Sabbin Kayayyakin Samfura Mai Kyau Synephrine Hydrochloride Foda

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Lokacin aikawa: Yuli-18-2025